SCHEMBL29907698

SCHEMBL29907698

Cc1ccc(-c2nc(N)c(C(=O)O)nc2-c2ccc(=O)n(C)c2)o1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.47
ADORA1 P30542 9/20 0.47
ADORA3 P0DMS8 1/20 0.47
ADORA2B P29275 3/20 0.43
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
RECQL P46063 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22552045 1.00 ADORA2A (0.47) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL22579112 0.89 ADORA2A (0.49) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL4584433 0.83 ADORA2A (0.56) ADORA2AADORA1ADORA2B
SCHEMBL29907718 0.82 ADORA2A (0.60) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL22552057 0.82 ADORA2A (0.60) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL4584998 0.82 ADORA2A (0.57) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL29987316 0.81 ADORA2A (0.65) ADORA2AADORA1ADORA2B
SCHEMBL4585883 0.81 ADORA2A (0.65) ADORA2AADORA1ADORA2B
SCHEMBL22579156 0.81 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL22551818 0.80 ADORA2A (0.78) ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2024-05-03 CN disclosed
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed