SCHEMBL29907718

SCHEMBL29907718

Cc1cc(-c2nc(C(=O)O)c(N)nc2-c2ccc(C)o2)cc(C)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.60
ADORA1 P30542 8/20 0.60
KAT8 Q9H7Z6 1/20 0.39
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 5/20 0.38
MAPT P10636 4/20 0.38
MEN1 O00255 2/20 0.38
POLB P06746 2/20 0.38
RECQL P46063 2/20 0.38
KMT2A Q03164 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
USP2 O75604 1/20 0.38
ADORA2B P29275 4/20 0.37
GLA P06280 2/20 0.36
HPGD P15428 2/20 0.36
PKM P14618 2/20 0.36
NR4A1 P22736 1/20 0.36
PPARG P37231 1/20 0.36
MCL1 Q07820 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22552057 1.00 ADORA2A (0.60) ADORA2AADORA1KAT8KDM4EALDH1A1
SCHEMBL22551849 0.88 ADORA2A (0.66) ADORA2AADORA1KDM4EALDH1A1MAPT
SCHEMBL22552045 0.82 ADORA2A (0.47) ADORA2AADORA1KDM4EALDH1A1MAPT
SCHEMBL29907698 0.82 ADORA2A (0.47) ADORA2AADORA1KDM4EALDH1A1MAPT
SCHEMBL21722434 0.81 ADORA2A (0.56) ADORA2AADORA1ADORA2B
SCHEMBL21722501 0.78 ADORA2A (0.57) ADORA2AADORA1ADORA2BADORA3
SCHEMBL29906757 0.78 ADORA2A (0.69) ADORA2AADORA1ADORA2BADORA3
SCHEMBL22552043 0.78 ADORA2A (0.69) ADORA2AADORA1ADORA2BADORA3
SCHEMBL22551864 0.76 ADORA2A (1.00) ADORA2AADORA1KDM4EALDH1A1MAPT
SCHEMBL29906683 0.76 ADORA2A (1.00) ADORA2AADORA1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2024-05-03 CN disclosed
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed