SCHEMBL29909155

SCHEMBL29909155

CNc1cccc(C(=O)Nc2ccccc2)c1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.67
POLB P06746 2/20 0.67
HDAC1 Q13547 1/20 0.67
HDAC2 Q92769 1/20 0.67
HDAC8 Q9BY41 1/20 0.67
HDAC6 Q9UBN7 1/20 0.67
KCNK3 O14649 4/20 0.65
KCNK9 Q9NPC2 4/20 0.65
RAB9A P51151 3/20 0.64
NPC1 O15118 3/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
SIRT1 Q96EB6 2/20 0.62
MEN1 O00255 6/20 0.61
PKM P14618 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
LMNA P02545 1/20 0.59
KDM4E B2RXH2 1/20 0.59
KCNH2 Q12809 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13001967 1.00 KMT2A (0.67) KMT2APOLBHDAC1HDAC2HDAC8
SCHEMBL23577148 0.89 KCNK3 (0.82) KMT2APOLBKCNK3KCNK9RAB9A
SCHEMBL17013407 0.87 KCNK3 (0.69) KMT2APOLBHDAC1HDAC2HDAC8
SCHEMBL11316890 0.87 PTGS1 (0.61) KMT2APOLBHDAC1HDAC2HDAC8
SCHEMBL8374911 0.87 HDAC1 (0.85) KMT2APOLBHDAC1HDAC2HDAC8
SCHEMBL15998541 0.85 HDAC1 (0.71) KMT2APOLBHDAC1HDAC2HDAC8
SCHEMBL19829331 0.85 MEN1 (0.67) KMT2APOLBHDAC1HDAC2HDAC8
SCHEMBL2685329 0.84 KCNK9 (0.67) KMT2APOLBHDAC8HDAC6KCNK3
SCHEMBL8940247 0.84 KCNK3 (0.72) KMT2APOLBHDAC1HDAC2HDAC8
SCHEMBL7151866 0.84 KMT2A (0.73) KMT2APOLBHDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12054490-B2 Diacylglycerol kinase modulating compounds GILEAD SCIENCES, INC. (US) 2024-08-06 US disclosed
CN-118324767-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2024-07-12 CN disclosed
CN-115362003-A Diacylglycerol kinase modulating compounds 卡尔那生物科学株式会社 2022-11-18 CN disclosed
EP-4081305-A1 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS Carna Biosciences, Inc. (JP) 2022-11-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12054490-B2 Diacylglycerol kinase modulating compounds DGKG, DGKB, DGKK KMT2A 2566/4885POLB 3027/4885HDAC1 1296/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.