Formic Acid

Formic Acid

SCHEMBL29911539

COCCOCCn1cc(NC(=O)c2cccc(-c3ccnc(C)c3)n2)c(-c2ccccn2)n1.O=CO

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 19/20 0.48
KCNH2 Q12809 2/20 0.42
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30261441 0.97 IRAK4 (0.50) IRAK4KCNH2CNR2
SCHEMBL20086065 0.97 IRAK4 (0.50) IRAK4KCNH2CNR2
Formic Acid SCHEMBL28976193 0.91 IRAK4 (0.47) IRAK4KCNH2
Formic Acid SCHEMBL30062335 0.89 IRAK4 (0.40) IRAK4
SCHEMBL30261532 0.89 IRAK4 (0.49) IRAK4KCNH2CNR2
SCHEMBL20086024 0.89 IRAK4 (0.49) IRAK4KCNH2CNR2
Formic Acid SCHEMBL29911777 0.88 IRAK4 (0.45) IRAK4KCNH2
SCHEMBL30051809 0.88 IRAK4 (0.50) IRAK4KCNH2
SCHEMBL20086023 0.88 IRAK4 (0.50) IRAK4KCNH2
Formic Acid SCHEMBL29911549 0.86 IRAK4 (0.50) IRAK4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115531387-A Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-12-30 CN claimed
CN-110234637-B Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-11-01 CN claimed
CN-110234637-B Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-11-01 CN disclosed