SCHEMBL29911712

SCHEMBL29911712

Cc1ccc(C(=O)Nc2cn(C)nc2-c2cnccn2)nc1-c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 13/20 0.56
ATR Q13535 2/20 0.41
ABL1 P00519 4/20 0.41
BCR P11274 4/20 0.41
PDGFRB P09619 3/20 0.41
EGFR P00533 2/20 0.41
PRKCA P17252 2/20 0.41
PDGFRA P16234 2/20 0.41
KCNH2 Q12809 1/20 0.41
PIM1 P11309 2/20 0.40
ESYT2 A0FGR8 1/20 0.40
HACL2 A1L0T0 1/20 0.40
NBAS A2RRP1 1/20 0.40
GTPBP10 A4D1E9 1/20 0.40
CNOT1 A5YKK6 1/20 0.40
TBKBP1 A7MCY6 1/20 0.40
AGPS O00116 1/20 0.40
ACOT7 O00154 1/20 0.40
MYO1F O00160 1/20 0.40
SNAP23 O00161 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29911867 0.91 IRAK4 (0.58) IRAK4ATRABL1BCRPDGFRB
SCHEMBL29911734 0.89 IRAK4 (0.52) IRAK4ATRABL1BCRPDGFRB
SCHEMBL20086030 0.87 IRAK4 (0.70) IRAK4KCNH2
SCHEMBL30261665 0.87 IRAK4 (0.70) IRAK4KCNH2
SCHEMBL28976258 0.86 IRAK4 (0.54) IRAK4ATRABL1BCRPDGFRB
SCHEMBL29911657 0.83 IRAK4 (0.49) IRAK4ABL1BCRPDGFRBEGFR
Hydrochloric Acid SCHEMBL29911751 0.83 IRAK4 (0.49) IRAK4ABL1BCRPDGFRBEGFR
SCHEMBL29911864 0.82 IRAK4 (0.53) IRAK4ABL1BCRPIM1PIM3
SCHEMBL29911831 0.81 IRAK4 (0.57) IRAK4ATRKCNH2HDAC1HDAC2
SCHEMBL29911856 0.81 IRAK4 (0.52) IRAK4ABL1BCRPIM1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115531387-A Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-12-30 CN claimed
CN-110234637-B Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-11-01 CN claimed
CN-115531387-A Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-12-30 CN disclosed
CN-110234637-B Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-11-01 CN disclosed