SCHEMBL29911734

SCHEMBL29911734

CC(=O)Nc1ccc(C(=O)Nc2cn(C)nc2-c2cnccn2)nc1-c1cccnc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 11/20 0.52
PIK3CA P42336 1/20 0.40
PIK3CG P48736 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
CYP1A2 P05177 1/20 0.39
ATR Q13535 1/20 0.39
PIM1 P11309 1/20 0.39
PIM3 Q86V86 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
ABL1 P00519 1/20 0.38
PDGFRB P09619 1/20 0.38
BCR P11274 1/20 0.38
PDGFRA P16234 1/20 0.38
KCNH2 Q12809 1/20 0.38
AURKA O14965 1/20 0.38
CSNK1D P48730 1/20 0.37
CSNK1E P49674 1/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29911712 0.89 IRAK4 (0.56) IRAK4ATRPIM1PIM3PIM2
SCHEMBL30261665 0.85 IRAK4 (0.70) IRAK4KCNH2
SCHEMBL20086030 0.85 IRAK4 (0.70) IRAK4KCNH2
SCHEMBL29911659 0.81 IRAK4 (0.52) IRAK4KCNH2JAK2JAK1
SCHEMBL29911867 0.80 IRAK4 (0.58) IRAK4ATRABL1PDGFRBBCR
SCHEMBL29911831 0.80 IRAK4 (0.57) IRAK4ATRKCNH2
SCHEMBL29911731 0.80 IRAK4 (0.55) IRAK4ATRPIM1PIM3PIM2
SCHEMBL28976258 0.79 IRAK4 (0.54) IRAK4ATRABL1PDGFRBBCR
SCHEMBL20089040 0.79 IRAK4 (0.54) IRAK4KCNH2
SCHEMBL29911961 0.78 IRAK4 (0.53) IRAK4ATRABL1BCRJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115531387-A Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-12-30 CN claimed
CN-110234637-B Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-11-01 CN claimed
CN-115531387-A Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-12-30 CN disclosed
CN-110234637-B Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-11-01 CN disclosed