SCHEMBL29912914

SCHEMBL29912914

COc1ccccc1-c1c(C(=O)O)c2nccnc2n1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
RAB9A P51151 2/20 0.40
EGLN1 Q9GZT9 1/20 0.40
NPC1 O15118 1/20 0.40
ATM Q13315 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA4 P48058 1/20 0.38
DHODH Q02127 2/20 0.38
HSD11B1 P28845 1/20 0.37
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27157885 1.00 CA12 (0.42) CA12CA1CA2CA7CA9
SCHEMBL29913278 0.83 MAPT (0.38) HPGDHSD17B10GRIA2GRIA4DHODH
SCHEMBL27157865 0.83 MAPT (0.38) HPGDHSD17B10GRIA2GRIA4DHODH
SCHEMBL6485737 0.80 CYP1A2 (0.42) CA1CA2ALDH1A1KDM4EHPGD
SCHEMBL29912955 0.80 CYP1A2 (0.42) CA1CA2ALDH1A1KDM4EHPGD
SCHEMBL30785435 0.79 GAA (0.38) ALDH1A1HPGDKMT2A
SCHEMBL27158658 0.79 GAA (0.38) ALDH1A1HPGDKMT2A
SCHEMBL29913098 0.74 KDM5A (0.43) KDM4EGRIA2GRIA4DHODHKMT2A
SCHEMBL9177751 0.74 EGFR (0.51) CA12CA1CA2CA7CA9
SCHEMBL27157832 0.74 KDM5A (0.43) KDM4EGRIA2GRIA4DHODHKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4329881-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF Vanqua Bio, Inc. (US) 2024-03-06 EP disclosed
CN-117642404-A Small molecule modulators of glucocerebrosidase activity and uses thereof 凡况生化公司 2024-03-01 CN disclosed
WO-2022232383-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2022-11-03 WO disclosed