SCHEMBL29914718

SCHEMBL29914718

COc1cnc(-c2cccc(O)c2)nc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
HSD17B1 P14061 6/20 0.54
HSD17B2 P37059 6/20 0.54
FYN P06241 5/20 0.48
HSD17B13 Q7Z5P4 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
BMPR1A P36894 1/20 0.44
TGFBR1 P36897 1/20 0.44
ACVRL1 P37023 1/20 0.44
ACVR1 Q04771 1/20 0.44
ABL1 P00519 2/20 0.44
BCR P11274 2/20 0.44
METAP2 P50579 1/20 0.44
ABCB1 P08183 1/20 0.44
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21228226 1.00 DYRK1A (0.54) DYRK1ACLK4HSD17B1HSD17B2FYN
SCHEMBL2222925 0.83 FYN (0.53) HSD17B1HSD17B2FYNHSD17B13CYP3A4
SCHEMBL27807278 0.83 DYRK1A (0.69) DYRK1ACLK4FYNCYP3A4CYP2C9
SCHEMBL27773721 0.81 CYP3A4 (0.58) HSD17B1HSD17B2FYNHSD17B13CYP3A4
SCHEMBL29786794 0.81 CLK4 (0.56) DYRK1ACLK4CYP3A4CYP2C9METAP2
SCHEMBL28810989 0.81 CLK4 (0.56) DYRK1ACLK4CYP3A4CYP2C9METAP2
SCHEMBL2221994 0.79 CLK4 (0.54) DYRK1ACLK4FYNCYP3A4ABCG2
SCHEMBL3389945 0.79 CLK4 (0.54) DYRK1ACLK4CYP3A4CYP2C9ABL1
SCHEMBL3219419 0.79 HSD17B1 (0.49) HSD17B1HSD17B2HSD17B13
SCHEMBL22310395 0.79 FYN (0.51) DYRK1ACLK4FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111094300-B Benzo-heteroaryl derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-09-16 CN disclosed