SCHEMBL29915324

SCHEMBL29915324

CCOP(=O)(Cc1cc(-c2cccc(Cl)c2)nn1Cc1ccc(OC)cc1)OCC

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.43
TP53 P04637 3/20 0.43
KDR P35968 1/20 0.40
EPHB4 P54760 1/20 0.40
TEK Q02763 1/20 0.40
HDAC1 Q13547 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
MAPK1 P28482 1/20 0.39
MAPK10 P53779 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GCGR P47871 1/20 0.38
NPBWR1 P48145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29915423 0.89 MAPT (0.46) MAPTHDAC1SMN1; SMN2MEN1KMT2A
SCHEMBL29915381 0.88 MAPT (0.41) MAPTTP53HDAC1SMN1; SMN2MEN1
SCHEMBL20600063 0.87 MAPT (0.45) MAPTTP53KDREPHB4TEK
SCHEMBL29915468 0.87 PTGDR (0.42) MAPTSMN1; SMN2MAPK1MEN1KMT2A
SCHEMBL29915480 0.84 TP53 (0.44) MAPTTP53MAPK1MAPK10GCGR
SCHEMBL29915535 0.84 MAPT (0.41) MAPTHDAC1SMN1; SMN2MEN1KMT2A
SCHEMBL29915488 0.83 MAPT (0.42) MAPTTP53SMN1; SMN2MEN1KMT2A
SCHEMBL22613601 0.82 MAPT (0.44) MAPTTP53KDREPHB4TEK
SCHEMBL22613652 0.81 MAPT (0.44) MAPTTP53KDREPHB4TEK
SCHEMBL22613710 0.76 MAPT (0.45) MAPTTP53HDAC1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11440922-B2 Heterocyclylmethylidene derivatives and their use as modulators of mGluR5 receptors Recordati Industria Chimica e Farmacentica S.p.A. (IT) 2022-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11440922-B2 Heterocyclylmethylidene derivatives and their use as modulators of mGluR5 receptors GRM5, GRIK5, GRM2 MAPT 361/4885TP53 4499/4885KDR 3892/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.