SCHEMBL29917310

SCHEMBL29917310

COc1cccc(-c2ccc(C(=O)NS(=O)(=O)c3cccc(N)n3)c(Oc3c(C)cc(C)cc3C)n2)n1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 10/20 0.35
SCN5A Q14524 1/20 0.34
PDCD1LG2 Q9BQ51 5/20 0.33
CD274 Q9NZQ7 5/20 0.33
FLT1 P17948 2/20 0.33
FLT4 P35916 2/20 0.33
KDR P35968 2/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
PTGES2 Q9H7Z7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17649011 1.00 SCN9A (0.35) SCN9ASCN5APDCD1LG2CD274FLT1
SCHEMBL17647916 0.92 RAB9A (0.39) SCN9ASCN5AFLT1FLT4KDR
SCHEMBL29917313 0.92 RAB9A (0.39) SCN9ASCN5AFLT1FLT4KDR
SCHEMBL19440522 0.91 SCN9A (0.34) SCN9ASCN5AFLT1FLT4KDR
SCHEMBL29918019 0.91 MAPT (0.35) SCN9ASCN5APDCD1LG2CD274FLT1
SCHEMBL17648396 0.91 MAPT (0.35) SCN9ASCN5APDCD1LG2CD274FLT1
SCHEMBL17648558 0.90 EGFR (0.36) SCN9ASCN5APDCD1LG2CD274FLT1
SCHEMBL29916753 0.90 EGFR (0.36) SCN9ASCN5APDCD1LG2CD274FLT1
SCHEMBL17648222 0.90 CD274 (0.37) SCN9ASCN5APDCD1LG2CD274NPC1
SCHEMBL29916237 0.90 CD274 (0.37) SCN9ASCN5APDCD1LG2CD274NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3798214-B1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2022-09-14 EP claimed