SCHEMBL29917657

SCHEMBL29917657

Cc1cc(C)c(Oc2nc(-c3ccccn3)ccc2C(=O)NS(=O)(=O)c2cccc(N)n2)c(C)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.38
MAPT P10636 4/20 0.38
POLB P06746 4/20 0.38
LMNA P02545 3/20 0.38
CCR6 P51684 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KMT2A Q03164 6/20 0.37
KDM4E B2RXH2 5/20 0.37
ADORA3 P0DMS8 3/20 0.37
MEN1 O00255 4/20 0.36
RXFP1 Q9HBX9 1/20 0.36
P4HTM Q9NXG6 1/20 0.36
KDM4A O75164 2/20 0.35
KDM4B O94953 2/20 0.35
KDM5B Q9UGL1 2/20 0.35
KDM5C P41229 1/20 0.35
HPGD P15428 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
USP2 O75604 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17648540 1.00 ALDH1A1 (0.38) ALDH1A1MAPTPOLBLMNACCR6
SCHEMBL29916466 0.91 FLT1 (0.35) ADORA3EGFR
SCHEMBL17649569 0.91 FLT1 (0.35) ADORA3EGFR
SCHEMBL29917943 0.90 SCN9A (0.35) EGFR
SCHEMBL17646908 0.90 SCN9A (0.35) EGFR
SCHEMBL17648558 0.90 EGFR (0.36) EGFR
SCHEMBL29916753 0.90 EGFR (0.36) EGFR
SCHEMBL17647665 0.89 ALDH1A1 (0.36) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL29916556 0.89 ALDH1A1 (0.36) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL29916838 0.88 SCN9A (0.36) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3798214-B1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2022-09-14 EP claimed