SCHEMBL29918458

SCHEMBL29918458

COc1cc(Nc2ncc(C(N)=O)cn2)cc(OC)c1

nearest known ligand 0.72

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 5/20 0.72
HDAC1 Q13547 5/20 0.72
HDAC2 Q92769 5/20 0.72
HDAC6 Q9UBN7 5/20 0.72
SYK P43405 6/20 0.53
PLAU P00749 1/20 0.49
HPGDS O60760 1/20 0.47
VNN1 O95497 2/20 0.46
CSF1R P07333 1/20 0.46
ZAP70 P43403 1/20 0.44
KARS1 Q15046 1/20 0.44
NNMT P40261 1/20 0.44
LCK P06239 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730352 0.84 HDAC1 (1.00) HDAC3HDAC1HDAC2HDAC6
SCHEMBL4485439 0.82 SYK (0.59) HDAC3HDAC1HDAC2HDAC6SYK
SCHEMBL2103980 0.77 AURKA (0.70) SYK
SCHEMBL14658780 0.73 MAPK8 (0.74) SYKZAP70
SCHEMBL10975772 0.73 HDAC3 (0.60) HDAC3HDAC1HDAC2HDAC6SYK
SCHEMBL8739793 0.72 HDAC3 (1.00) HDAC3HDAC1HDAC2HDAC6
SCHEMBL4487993 0.72 HDAC6 (0.68) HDAC3HDAC1HDAC2HDAC6SYK
SCHEMBL894796 0.72 PARP1 (0.64) PLAUHPGDS
SCHEMBL30033167 0.72 SYK (0.54) HDAC3HDAC1HDAC2HDAC6SYK
SCHEMBL3634270 0.71 HDAC3 (0.74) HDAC3HDAC1HDAC2HDAC6SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115073467-B Pyrimidine imidazole compound, and pharmaceutical composition and application thereof 中国科学院上海药物研究所 2024-03-15 CN disclosed
CN-115073467-A Pyrimido imidazole compound and medicinal composition and application thereof 中国科学院上海药物研究所 2022-09-20 CN disclosed