SCHEMBL29922290

SCHEMBL29922290

NC(=O)c1cnc(Cl)nc1N[C@H](CO)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 14/20 0.56
AURKA O14965 11/20 0.56
IRAK4 Q9NWZ3 4/20 0.55
JAK3 P52333 1/20 0.55
MAP4K1 Q92918 3/20 0.52
MAP4K3 Q8IVH8 2/20 0.52
AURKB Q96GD4 3/20 0.45
EGFR P00533 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28459567 0.90 IRAK4 (0.51) RPS6KB1AURKAIRAK4JAK3MAP4K1
SCHEMBL29922002 0.90 IRAK4 (0.51) RPS6KB1AURKAIRAK4JAK3MAP4K1
SCHEMBL22773044 0.90 IRAK4 (0.51) RPS6KB1AURKAIRAK4JAK3MAP4K1
SCHEMBL29922295 0.89 AURKA (0.47) RPS6KB1AURKAIRAK4JAK3MAP4K1
SCHEMBL24612853 0.83 MAP4K1 (0.56) RPS6KB1AURKAIRAK4MAP4K1MAP4K3
SCHEMBL22785699 0.83 MAP4K1 (0.56) RPS6KB1AURKAIRAK4MAP4K1MAP4K3
SCHEMBL30504131 0.83 MAP4K1 (0.56) RPS6KB1AURKAIRAK4MAP4K1MAP4K3
SCHEMBL30431469 0.83 MAP4K1 (0.56) RPS6KB1AURKAIRAK4MAP4K1MAP4K3
SCHEMBL913833 0.82 AURKA (0.54) RPS6KB1AURKAAURKBEGFR
SCHEMBL14670573 0.82 EGFR (0.46) RPS6KB1AURKAEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022188735-A1 HETEROCYCLIC COMPOUNDS AS HPK1 INHIBITORS GUANGDONG NEWOPP BIOPHARMACEUTICALS CO., LTD. (CN) 2022-09-15 WO disclosed