SCHEMBL29923403

SCHEMBL29923403

c1ccc2c(-c3nccc4ccccc34)nccc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 2/20 0.60
CYP2A6 P11509 2/20 0.60
F12 P00748 1/20 0.60
NCF1 P14598 1/20 0.60
NOS3 P29474 1/20 0.60
NOS1 P29475 1/20 0.60
NOS2 P35228 1/20 0.60
BACE1 P56817 1/20 0.60
MAPT P10636 5/20 0.58
NPC1 O15118 4/20 0.58
RAB9A P51151 4/20 0.58
KDM4E B2RXH2 4/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
KMT2A Q03164 2/20 0.58
GLA P06280 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
GPR55 Q9Y2T6 1/20 0.53
PLG P00747 1/20 0.48
ALDH1A1 P00352 3/20 0.48
HSD17B10 Q99714 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL199273 1.00 PLAU (0.60) PLAUCYP2A6F12NCF1NOS3
SCHEMBL30522769 0.97 PLAU (0.58) PLAUCYP2A6F12NCF1NOS3
SCHEMBL13978866 0.90 PLAU (0.56) PLAUCYP2A6F12NCF1NOS3
SCHEMBL12223316 0.90 PLAU (0.56) PLAUCYP2A6F12NCF1NOS3
SCHEMBL12112873 0.88 MAPT (0.58) PLAUCYP2A6F12NCF1NOS3
SCHEMBL4500979 0.87 KDM4E (0.53) PLAUCYP2A6F12NCF1NOS3
Dipyridyl SCHEMBL4596384 0.87 KDM4E (0.56) PLAUCYP2A6F12NCF1NOS3
SCHEMBL50715 0.86 KDM4E (0.66) PLAUCYP2A6F12NCF1NOS3
SCHEMBL29398625 0.86 KDM4E (0.66) PLAUCYP2A6F12NCF1NOS3
SCHEMBL24663020 0.84 MAPT (0.50) PLAUCYP2A6F12NCF1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116874421-A Method for synthesizing 1,1' -biisoquinoline derivative from 2, 2-dimethyl-4, 5-diaryl-2H-imidazole 桂林理工大学 2023-10-13 CN claimed
CN-116621777-A Method for synthesizing 1,1' -biisoquinoline oxynitride 桂林理工大学 2023-08-22 CN claimed
CN-116874421-A Method for synthesizing 1,1' -biisoquinoline derivative from 2, 2-dimethyl-4, 5-diaryl-2H-imidazole 桂林理工大学 2023-10-13 CN disclosed
CN-116874421-A Method for synthesizing 1,1' -biisoquinoline derivative from 2, 2-dimethyl-4, 5-diaryl-2H-imidazole 桂林理工大学 2023-10-13 CN disclosed
CN-116874421-A Method for synthesizing 1,1' -biisoquinoline derivative from 2, 2-dimethyl-4, 5-diaryl-2H-imidazole 桂林理工大学 2023-10-13 CN disclosed
CN-116621777-A Method for synthesizing 1,1' -biisoquinoline oxynitride 桂林理工大学 2023-08-22 CN disclosed
CN-116621777-A Method for synthesizing 1,1' -biisoquinoline oxynitride 桂林理工大学 2023-08-22 CN disclosed
CN-116621777-A Method for synthesizing 1,1' -biisoquinoline oxynitride 桂林理工大学 2023-08-22 CN disclosed
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed