SCHEMBL29923677

SCHEMBL29923677

Cc1cc(N)c(C=O)c(Br)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
KDM4E B2RXH2 2/20 0.38
ERN1 O75460 4/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
GAA P10253 1/20 0.34
PRKDC P78527 1/20 0.34
CYP3A4 P08684 3/20 0.33
CA1 P00915 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
TSHR P16473 2/20 0.33
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33
ALOX15 P16050 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALPG P10696 1/20 0.33
ALDH2 P05091 1/20 0.32
ALDH3A1 P30838 1/20 0.32
CA2 P00918 2/20 0.31
CA9 Q16790 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL304092 0.84 ERN1 (0.41) ALDH1A1KDM4EERN1LMNAMAPT
SCHEMBL18553998 0.78 ERN1 (0.42) ALDH1A1ERN1PRKDCCYP3A4CA1
SCHEMBL21130264 0.75 ALDH1A1 (0.37) ALDH1A1KDM4EERN1LMNAMAPT
SCHEMBL12581708 0.75 CYP3A4 (0.46) ALDH1A1ERN1MAPTPRKDCCYP3A4
SCHEMBL31189003 0.75 MEN1 (0.37) ALDH1A1KDM4EERN1LMNAMAPT
SCHEMBL16207565 0.75 ERN1 (0.34) ALDH1A1ERN1LMNAMAPTPRKDC
SCHEMBL31353446 0.75 CA1 (0.33) ERN1LMNAGAAPRKDCCA1
SCHEMBL12581710 0.72 PRKDC (0.53) ALDH1A1KDM4EERN1LMNAMAPT
SCHEMBL31426082 0.72 ERN1 (0.33) ALDH1A1ERN1LMNAMAPTPRKDC
SCHEMBL22060773 0.71 CYP3A4 (0.36) ALDH1A1ERN1MAPTPRKDCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4334305-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2024-03-13 EP disclosed
WO-2022236101-A1 WDR5 INHIBITORS AND MODULATORS VANDERBILT UNIVERSITY (US) 2022-11-10 WO disclosed
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed