SCHEMBL29924339

SCHEMBL29924339

COc1cc(Cl)ccc1C1COc2cccc(Br)c2O1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
HTR2A P28223 2/20 0.37
MAPT P10636 2/20 0.37
TSHR P16473 2/20 0.37
ADRA1D P25100 5/20 0.36
ADRA1A P35348 5/20 0.36
ADRA1B P35368 5/20 0.36
CSF1R P07333 4/20 0.36
DPP4 P27487 1/20 0.35
HTR2C P28335 2/20 0.34
HTR1A P08908 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
CYP19A1 P11511 2/20 0.34
NPC1 O15118 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29150031 1.00 HTT (0.43) HTTHTR2AMAPTTSHRADRA1D
SCHEMBL29924327 0.85 PTGS1 (0.35) HTTHTR2ATSHRCSF1RDPP4
SCHEMBL29149833 0.85 PTGS1 (0.35) HTTHTR2ATSHRCSF1RDPP4
SCHEMBL29149759 0.85 PTGS1 (0.35) HTTHTR2ATSHRCSF1RDPP4
SCHEMBL29924595 0.85 PTGS1 (0.35) HTTHTR2ATSHRCSF1RDPP4
SCHEMBL24186456 0.82 HTR2A (0.37) HTTHTR2AMAPTHTR2CNPC1
SCHEMBL29924349 0.82 HTR2A (0.37) HTTHTR2AMAPTHTR2CNPC1
SCHEMBL23980833 0.82 HTR2A (0.37) HTTHTR2AMAPTHTR2CNPC1
SCHEMBL29924375 0.81 HTR2C (0.44) HTTHTR2CHTR1A
SCHEMBL29149862 0.81 HTR2C (0.44) HTTHTR2CHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed