SCHEMBL29928879

SCHEMBL29928879

c1ccc(Cn2ccc3ccccc32)nc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 4/20 0.53
CCND1 P24385 4/20 0.53
BRD4 O60885 2/20 0.53
KMT2A Q03164 3/20 0.51
SLC2A1 P11166 1/20 0.51
HTR6 P50406 1/20 0.50
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
GRIN1 Q05586 1/20 0.44
KCNH2 Q12809 1/20 0.44
GRIN2B Q13224 1/20 0.44
PLAU P00749 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
PKM P14618 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
GABRA1 P14867 1/20 0.43
GABRA5 P31644 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11225244 1.00 CDK4 (0.53) CDK4CCND1BRD4KMT2ASLC2A1
SCHEMBL13416068 0.84 CDK4 (0.59) CDK4CCND1KMT2AHTR6PLAU
SCHEMBL12542891 0.83 CDK4 (0.59) CDK4CCND1HTR2AHTR2C
SCHEMBL28690469 0.82 CDK4 (0.49) CDK4CCND1KMT2AHTR6PLAU
SCHEMBL916444 0.82 BRD4 (0.56) BRD4SLC2A1HTR6CYP1A2CYP2C9
SCHEMBL31661504 0.82 SLC2A1 (0.54) BRD4SLC2A1HTR6CYP1A2CYP2C9
SCHEMBL3507524 0.82 SLC2A1 (0.54) BRD4SLC2A1HTR6CYP1A2CYP2C9
SCHEMBL4035941 0.82 SLC2A1 (0.45) BRD4KMT2ASLC2A1CYP1A2CYP2C9
SCHEMBL17067797 0.82 BRD4 (0.56) BRD4SLC2A1CYP1A2CYP2C9CYP2C19
SCHEMBL28572469 0.78 BRD4 (0.47) BRD4SLC2A1HTR6CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113004188-B Indole derivative, preparation method and application 沈阳药科大学 2022-09-20 CN disclosed