SCHEMBL29929396

SCHEMBL29929396

O=C1C(=Cc2cc(Cl)ccc2Cl)CNCC1=Cc1cc(Cl)ccc1Cl

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK2 Q92630 3/20 0.65
PTP4A3 O75365 1/20 0.50
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
IKBKB O14920 6/20 0.47
RAF1 P04049 2/20 0.47
RPS6KB1 P23443 2/20 0.47
MAPK1 P28482 2/20 0.47
AKT1 P31749 2/20 0.47
AKT2 P31751 2/20 0.47
KDR P35968 2/20 0.47
PRKAG1 P54619 2/20 0.47
MAP2K1 Q02750 2/20 0.47
PRKAA1 Q13131 2/20 0.47
MAPK14 Q16539 2/20 0.47
NEK1 Q96PY6 2/20 0.47
PRKAB1 Q9Y478 2/20 0.47
ACHE P22303 2/20 0.43
PTGS2 P35354 1/20 0.43
BCHE P06276 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29929498 0.83 DYRK2 (0.61) DYRK2PTP4A3CRHBPCRHR2IKBKB
SCHEMBL29929309 0.83 IKBKB (0.61) DYRK2IKBKBRAF1RPS6KB1MAPK1
SCHEMBL29928652 0.80 IKBKB (0.61) DYRK2IKBKBRAF1RPS6KB1MAPK1
SCHEMBL29929418 0.79 DYRK2 (1.00) DYRK2IKBKBRAF1RPS6KB1MAPK1
SCHEMBL13036873 0.79 DYRK2 (1.00) DYRK2IKBKBRAF1RPS6KB1MAPK1
SCHEMBL7122621 0.79 DYRK2 (1.00) DYRK2IKBKBRAF1RPS6KB1MAPK1
SCHEMBL7122623 0.79 DYRK2 (1.00) DYRK2IKBKBRAF1RPS6KB1MAPK1
SCHEMBL13719949 0.74 IKBKB (0.67) DYRK2IKBKBACHEPTGS2BCHE
SCHEMBL13719950 0.74 IKBKB (0.67) DYRK2IKBKBACHEPTGS2BCHE
SCHEMBL23095004 0.74 IKBKB (0.56) DYRK2IKBKBRAF1RPS6KB1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232068-B Compound and preparation method and application thereof 北京中医药大学 2023-09-08 CN disclosed
CN-115232068-B Compound and preparation method and application thereof 北京中医药大学 2023-09-08 CN disclosed
CN-115232068-A Compound and preparation method and application thereof 北京中医药大学 2022-10-25 CN disclosed
CN-115232068-A Compound and preparation method and application thereof 北京中医药大学 2022-10-25 CN disclosed