SCHEMBL299338

SCHEMBL299338

Cc1nc(Br)sc1C(=O)NCCCn1ccnc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.61
SMN1; SMN2 Q16637 4/20 0.57
PKM P14618 1/20 0.57
NPC1 O15118 1/20 0.56
ALDH1A1 P00352 4/20 0.55
KMT2A Q03164 3/20 0.55
CYP19A1 P11511 1/20 0.55
MAPT P10636 1/20 0.55
TSHR P16473 1/20 0.55
MEN1 O00255 1/20 0.55
KDM4E B2RXH2 2/20 0.53
POLB P06746 2/20 0.53
LMNA P02545 1/20 0.53
HTT P42858 1/20 0.53
HSD17B10 Q99714 1/20 0.53
TP53 P04637 1/20 0.52
MAPK1 P28482 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5614303 0.85 NAMPT (0.58) NAMPTSMN1; SMN2PKMNPC1ALDH1A1
SCHEMBL774992 0.80 NAMPT (0.52) NAMPTSMN1; SMN2PKMALDH1A1KMT2A
SCHEMBL11087591 0.76 NAMPT (0.65) NAMPTSMN1; SMN2NPC1ALDH1A1KMT2A
SCHEMBL16227562 0.76 NAMPT (0.64) NAMPTSMN1; SMN2NPC1ALDH1A1CYP19A1
SCHEMBL21098369 0.74 SMN1; SMN2 (0.89) SMN1; SMN2NPC1ALDH1A1KMT2ACYP19A1
SCHEMBL12330491 0.74 MEN1 (0.70) NAMPTSMN1; SMN2NPC1ALDH1A1KMT2A
SCHEMBL13211944 0.74 SMN1; SMN2 (0.78) NAMPTSMN1; SMN2NPC1ALDH1A1KMT2A
SCHEMBL4770380 0.74 SMN1; SMN2 (0.78) SMN1; SMN2NPC1ALDH1A1KMT2ACYP19A1
SCHEMBL6398857 0.74 L3MBTL1 (0.68) NAMPTSMN1; SMN2NPC1ALDH1A1KMT2A
SCHEMBL9906905 0.73 MEN1 (0.65) NAMPTSMN1; SMN2NPC1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed