SCHEMBL29933932

SCHEMBL29933932

Nc1cncc(-c2ncccn2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.48
DYRK1B Q9Y463 2/20 0.45
DYRK1A Q13627 2/20 0.44
MEN1 O00255 3/20 0.42
PSIP1 O75475 1/20 0.42
AXL P30530 1/20 0.42
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
DDO Q99489 1/20 0.41
NTRK1 P04629 1/20 0.40
CYP11B2 P19099 2/20 0.38
CYP11B1 P15538 1/20 0.38
CLK2 P49760 1/20 0.37
CLK3 P49761 1/20 0.37
ADRB2 P07550 1/20 0.36
MAP4K4 O95819 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5027205 1.00 CYP2A6 (0.48) CYP2A6DYRK1BDYRK1AMEN1PSIP1
Hydrochloric Acid SCHEMBL23501615 0.98 CYP2A6 (0.47) CYP2A6DYRK1BDYRK1AMEN1PSIP1
Hydrochloric Acid SCHEMBL29933924 0.98 CYP2A6 (0.47) CYP2A6DYRK1BDYRK1AMEN1PSIP1
SCHEMBL17546483 0.77 ADRB2 (0.41) CYP2A6DYRK1AMEN1PSIP1AXL
SCHEMBL14955802 0.77 ADRB2 (0.41) CYP2A6DYRK1AMEN1PSIP1AXL
SCHEMBL15220476 0.76 CYP2A6 (0.56) CYP2A6DYRK1BDYRK1AMEN1PSIP1
SCHEMBL12117526 0.74 CYP2A6 (0.48) CYP2A6DYRK1ACYP11B2CYP11B1
SCHEMBL23501651 0.74 CYP2A6 (0.48) CYP2A6DYRK1BDYRK1AMEN1KDM4E
SCHEMBL5799279 0.74 PTK2 (0.52) CYP2A6MEN1KDM4EALDH1A1KMT2A
SCHEMBL23501621 0.74 CYP2A6 (0.48) CYP2A6MKNK1MKNK2CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119371371-A Compounds and compositions as PDGF receptor kinase inhibitors 日本新药株式会社 2025-01-28 CN disclosed
CN-115315421-B Compounds and compositions as PDGF receptor kinase inhibitors 日本新药株式会社 2024-12-03 CN disclosed
CN-115315421-A Compounds and compositions as PDGF receptor kinase inhibitors 日本新药株式会社 2022-11-08 CN disclosed