SCHEMBL29936015

SCHEMBL29936015

CN(C)c1cccc2c(S(=O)(=O)NC[C@H](N)C(=O)O)cccc12

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.55
HDAC10 Q969S8 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
HDAC5 Q9UQL6 1/20 0.55
F2 P00734 2/20 0.54
PRSS1 P07477 2/20 0.54
PRSS2 P07478 2/20 0.54
PRSS3 P35030 2/20 0.54
EDNRA P25101 6/20 0.52
CA2 P00918 1/20 0.51
GBA1 P04062 2/20 0.51
PTGS2 P35354 1/20 0.49
EPHX2 P34913 1/20 0.48
HDAC1 Q13547 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13911551 1.00 HDAC4 (0.55) HDAC4HDAC10HDAC6HDAC5F2
SCHEMBL869336 1.00 HDAC4 (0.55) HDAC4HDAC10HDAC6HDAC5F2
SCHEMBL29462219 1.00 HDAC4 (0.55) HDAC4HDAC10HDAC6HDAC5F2
SCHEMBL9163130 0.88 HDAC4 (0.58) HDAC4HDAC10HDAC6HDAC5F2
SCHEMBL14110615 0.88 HDAC4 (0.48) HDAC4HDAC10HDAC6HDAC5F2
SCHEMBL14110750 0.85 HDAC4 (0.55) HDAC4HDAC10HDAC6HDAC5F2
SCHEMBL13651429 0.85 HDAC4 (0.64) HDAC4HDAC10HDAC6HDAC5GBA1
SCHEMBL29358078 0.85 HDAC4 (0.64) HDAC4HDAC10HDAC6HDAC5GBA1
SCHEMBL597355 0.85 HDAC4 (0.64) HDAC4HDAC10HDAC6HDAC5GBA1
SCHEMBL18612351 0.82 EDNRA (0.59) HDAC4HDAC10HDAC6HDAC5F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025080877-A2 THERAPEUTIC PEPTIDES FREZENT BIOLOGICAL SOLUTIONS, INC. (US) 2025-04-17 WO disclosed
US-20240327850-A1 METHODS AND COMPOSITIONS FOR CONTROLLING RELEASE FACTOR ACTIVITY AND USES THEREOF OXFORD FINANCE LLC, AS COLLATERAL AGENT 2024-10-03 US disclosed
WO-2024086738-A2 COMPOSITIONS AND METHODS OF USE FOR INTEINS GRO BIOSCIENCES INC. (US) 2024-04-25 WO disclosed
WO-2022235825-A1 METHODS AND COMPOSITIONS FOR CONTROLLING RELEASE FACTOR ACTIVITY AND USES THEREOF Opentrons LabWorks Inc. (US) 2022-11-10 WO disclosed
WO-2022221576-A1 METHODS FOR CODON OPTIMIZATION AND USES THEREOF Opentrons LabWorks Inc. (US) 2022-10-20 WO disclosed