SCHEMBL29936657

SCHEMBL29936657

COc1ccc(-c2noc(-c3ccc(N)cc3)n2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 13/20 0.74
NPC1 O15118 12/20 0.74
MAPT P10636 10/20 0.74
SMN1; SMN2 Q16637 6/20 0.74
NR1H4 Q96RI1 3/20 0.74
NPSR1 Q6W5P4 2/20 0.74
S1PR1 P21453 1/20 0.74
HPGD P15428 4/20 0.61
KDM4E B2RXH2 4/20 0.61
NFKB1 P19838 3/20 0.61
NFKB2 Q00653 3/20 0.61
RELA Q04206 3/20 0.61
ALDH1A1 P00352 3/20 0.61
TP53 P04637 2/20 0.61
HSD17B10 Q99714 2/20 0.61
LMNA P02545 2/20 0.58
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
TPH1 P17752 2/20 0.57
PKM P14618 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16592531 1.00 RAB9A (0.74) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL6697420 0.85 NR1H4 (1.00) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL7291752 0.85 NR1H4 (1.00) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL12895918 0.85 RAB9A (0.76) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL13416230 0.84 NPC1 (1.00) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL3057492 0.84 RAB9A (0.74) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL26095707 0.84 RAB9A (1.00) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL3057134 0.84 RAB9A (0.74) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL16769354 0.83 NPC1 (0.68) RAB9ANPC1MAPTSMN1; SMN2NR1H4
SCHEMBL16592612 0.83 RAB9A (0.72) RAB9ANPC1MAPTSMN1; SMN2NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4304630-A1 SMALL MOLECULE ANTAGONISTS FOR THE RELAXIN-3/RXFP3 SYSTEM Research Triangle Institute (US) 2024-01-17 EP disclosed
WO-2022192126-A1 SMALL MOLECULE ANTAGONISTS FOR THE RELAXIN-3/RXFP3 SYSTEM RESEARCH TRIANGLE INSTITUTE (US) 2022-09-15 WO disclosed