SCHEMBL29936770

SCHEMBL29936770

Cc1ccc([C@@H](N)CC2CC2)cc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
OPRL1 P41146 1/20 0.45
CRHR1 P34998 2/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
ALDH1A1 P00352 5/20 0.35
LMNA P02545 4/20 0.34
KMT2A Q03164 4/20 0.34
MEN1 O00255 3/20 0.34
POLB P06746 2/20 0.34
HTT P42858 2/20 0.34
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CCR5 P51681 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL892427 1.00 OPRM1 (0.45) OPRM1OPRD1OPRK1OPRL1CRHR1
SCHEMBL5469779 1.00 OPRM1 (0.45) OPRM1OPRD1OPRK1OPRL1CRHR1
Hydrochloric Acid SCHEMBL28652117 0.98 OPRM1 (0.44) OPRM1OPRD1OPRK1OPRL1CRHR1
Hydrochloric Acid SCHEMBL28652116 0.98 OPRM1 (0.44) OPRM1OPRD1OPRK1OPRL1CRHR1
SCHEMBL25871714 0.85 HPGD (0.34) OPRM1OPRD1OPRK1OPRL1ALDH1A1
SCHEMBL24222041 0.84 OPRL1 (0.43) OPRM1OPRD1OPRK1OPRL1AKR1C3
SCHEMBL27549476 0.79 DPP4 (0.33)
SCHEMBL14981098 0.76 ANPEP (0.41) OPRM1OPRD1OPRK1OPRL1AKR1C3
SCHEMBL5407290 0.76 AKR1C3 (0.41) OPRM1OPRD1OPRK1OPRL1AKR1C3
SCHEMBL24262071 0.76 AKR1C3 (0.41) OPRM1OPRD1OPRK1OPRL1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115087647-A Synthetic method for preparing 4- (2-chloro-4-methoxy-5-methylphenyl) -N- [ (1S) -2-cyclopropyl-1- (3-fluoro-4-methylphenyl) ethyl ] -5-methyl-N-prop-2-alkynyl-1, 3-thiazol-2-amine 纽罗克里生物科学有限公司 2022-09-20 CN claimed
CN-116322668-A Synthetic method for preparing 4- (2-chloro-4-methoxy-5-methylphenyl) -N- [ (1S) -2-cyclopropyl-1- (3-fluoro-4-methylphenyl) ethyl ] -5-methyl-N-prop-2-ynyl-1, 3-thiazol-2-amine 纽罗克里生物科学有限公司 2023-06-23 CN disclosed
CN-115087647-A Synthetic method for preparing 4- (2-chloro-4-methoxy-5-methylphenyl) -N- [ (1S) -2-cyclopropyl-1- (3-fluoro-4-methylphenyl) ethyl ] -5-methyl-N-prop-2-alkynyl-1, 3-thiazol-2-amine 纽罗克里生物科学有限公司 2022-09-20 CN disclosed