SCHEMBL29937151

SCHEMBL29937151

COCOc1ccc2ccccc2c1Br

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.56
HPGD P15428 1/20 0.56
PRNP P04156 5/20 0.50
RXFP1 Q9HBX9 4/20 0.50
LMNA P02545 1/20 0.50
RAB9A P51151 4/20 0.49
TP53 P04637 1/20 0.49
MAPK1 P28482 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
MAPT P10636 4/20 0.49
NCEH1 Q6PIU2 4/20 0.49
NPC1 O15118 2/20 0.49
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 2/20 0.47
TSHR P16473 2/20 0.47
KMT2A Q03164 2/20 0.47
HTT P42858 1/20 0.47
ADRB2 P07550 1/20 0.47
POLB P06746 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7380732 1.00 SMN1; SMN2 (0.56) SMN1; SMN2HPGDPRNPRXFP1LMNA
SCHEMBL29625686 0.83 PRNP (0.50) SMN1; SMN2HPGDPRNPRXFP1LMNA
SCHEMBL23515145 0.83 PRNP (0.50) SMN1; SMN2HPGDPRNPRXFP1LMNA
SCHEMBL26622001 0.82 RAB9A (0.55) SMN1; SMN2HPGDPRNPRXFP1LMNA
SCHEMBL29820187 0.82 MAPT (0.63) SMN1; SMN2HPGDRAB9AMAPTALDH1A1
SCHEMBL1446528 0.82 MAPT (0.63) SMN1; SMN2HPGDRAB9AMAPTALDH1A1
SCHEMBL15287590 0.81 SMN1; SMN2 (0.36) SMN1; SMN2HPGDPRNPRXFP1LMNA
SCHEMBL12745123 0.81 MAPT (0.58) SMN1; SMN2HPGDPRNPRXFP1LMNA
SCHEMBL15285233 0.81 MAPT (0.47) SMN1; SMN2HPGDRAB9AMAPTNPC1
SCHEMBL8731312 0.81 NCEH1 (0.47) SMN1; SMN2HPGDRAB9AMAPK1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118812473-A Naphthyl-coumarin molecular probe and synthetic method and application thereof 达州中医药职业学院 2024-10-22 CN disclosed
EP-4322954-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT Merck Sharp & Dohme LLC (US) 2024-02-21 EP disclosed
EP-4087573-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2022-11-16 EP disclosed
WO-2022221739-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT MERCK SHARP & DOHME CORP. (US) 2022-10-20 WO disclosed