SCHEMBL29937291

SCHEMBL29937291

N#CCC12CCC(CNC1)N2C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.32
JAK2 O60674 2/20 0.31
JAK1 P23458 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29937133 0.81
SCHEMBL25324095 0.80 JAK1 (0.36) JAK2JAK1
SCHEMBL3822469 0.77
SCHEMBL25211808 0.77 DPP4 (0.30)
SCHEMBL25415541 0.77 DPP4 (0.30)
SCHEMBL25413586 0.75
SCHEMBL30520607 0.75
SCHEMBL25414126 0.75
SCHEMBL30520497 0.75
SCHEMBL30520662 0.74 DPP4 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4322954-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT Merck Sharp & Dohme LLC (US) 2024-02-21 EP disclosed
WO-2022221739-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT MERCK SHARP & DOHME CORP. (US) 2022-10-20 WO disclosed