SCHEMBL29937394

SCHEMBL29937394

[2H]Cc1cc2[nH]ncc2c(Br)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.41
TDO2 P48775 1/20 0.41
METAP2 P50579 10/20 0.40
NOS1 P29475 6/20 0.36
AXL P30530 2/20 0.36
CYP1A2 P05177 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
PTPN6 P29350 1/20 0.33
DYRK1A Q13627 3/20 0.33
CSNK2A1 P68400 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21195949 0.88 IDO1 (0.44) IDO1TDO2METAP2NOS1AXL
SCHEMBL30007907 0.88 IDO1 (0.44) IDO1TDO2METAP2NOS1AXL
SCHEMBL21195941 0.79 IDO1 (0.46) IDO1TDO2METAP2NOS1AXL
SCHEMBL29804020 0.79 IDO1 (0.46) IDO1TDO2METAP2NOS1AXL
SCHEMBL30959639 0.77 IDO1 (0.44) IDO1TDO2METAP2NOS1AXL
SCHEMBL31642846 0.76 IDO1 (0.43) IDO1TDO2METAP2NOS1AXL
SCHEMBL21196002 0.76 IDO1 (0.43) IDO1TDO2METAP2NOS1AXL
SCHEMBL30187208 0.76 IDO1 (0.43) IDO1TDO2METAP2NOS1AXL
SCHEMBL21196238 0.74 IDO1 (0.48) IDO1TDO2METAP2NOS1AXL
SCHEMBL30410207 0.73 IDO1 (0.47) IDO1TDO2METAP2NOS1AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4322954-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT Merck Sharp & Dohme LLC (US) 2024-02-21 EP disclosed
WO-2022221739-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT MERCK SHARP & DOHME CORP. (US) 2022-10-20 WO disclosed