SCHEMBL29939082

SCHEMBL29939082

O=C(Nc1cnc(F)cc1N1CCOCC1)c1ccnc(Nc2cccc(OC(F)(F)F)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 4/20 0.49
GSK3B P49841 4/20 0.49
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CTSS P25774 1/20 0.47
CTSK P43235 1/20 0.47
BRAF P15056 3/20 0.44
AKT1 P31749 1/20 0.43
MET P08581 1/20 0.43
EGFR P00533 1/20 0.43
ITK Q08881 1/20 0.43
SYK P43405 2/20 0.42
RAF1 P04049 1/20 0.42
PIM1 P11309 1/20 0.42
IGF1R P08069 1/20 0.42
BTK Q06187 1/20 0.42
CSF1R P07333 1/20 0.41
DAPK1 P53355 1/20 0.41
MTOR P42345 1/20 0.41
SMG1 Q96Q15 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20190085 1.00 GSK3A (0.49) GSK3AGSK3BCTSLCTSBCTSS
SCHEMBL20205183 0.87 GSK3A (0.53) GSK3AGSK3BBTKMTORSMG1
SCHEMBL20204994 0.83 GSK3A (0.54) GSK3AGSK3BSYKPIM1BTK
SCHEMBL29939489 0.82 GSK3A (0.49) GSK3AGSK3BSYKPIM1BTK
SCHEMBL20205219 0.82 GSK3A (0.49) GSK3AGSK3BSYKPIM1BTK
SCHEMBL20189914 0.80 JAK2 (0.55) GSK3AGSK3BSYKPIM1IGF1R
SCHEMBL20205173 0.78 MAPK1 (0.52) GSK3AGSK3BIRAK4
SCHEMBL29939117 0.78 MAPK1 (0.52) GSK3AGSK3BIRAK4
SCHEMBL20204972 0.78 TSHR (0.51) GSK3AGSK3BIRAK4
SCHEMBL29939856 0.78 TSHR (0.51) GSK3AGSK3BIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110545817-B GSK-3 inhibitors 百时美施贵宝公司 2022-11-15 CN disclosed