SCHEMBL29939620

SCHEMBL29939620

O=C(Nc1nc2c(Br)ncc(N3CCOCC3)c2s1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.51
ADORA2A P29274 3/20 0.49
ADORA1 P30542 3/20 0.49
ALDH1A1 P00352 3/20 0.48
NPC1 O15118 1/20 0.48
ATM Q13315 1/20 0.48
RAB9A P51151 2/20 0.46
POLB P06746 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
KDM4E B2RXH2 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
STAT3 P40763 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SCN9A Q15858 1/20 0.43
KDR P35968 1/20 0.43
ADORA3 P0DMS8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20702439 1.00 LRRK2 (0.51) LRRK2ADORA2AADORA1ALDH1A1NPC1
SCHEMBL3049478 0.82 LRRK2 (0.53) LRRK2ADORA2AADORA1ALDH1A1NPC1
SCHEMBL20702500 0.80 LRRK2 (0.59) LRRK2ADORA2AADORA1ALDH1A1NPC1
SCHEMBL3047856 0.79 ADORA2A (0.69) ADORA2AADORA1MEN1KMT2AADORA3
SCHEMBL2320399 0.77 ALDH1A1 (0.58) LRRK2ALDH1A1NPC1ATMRAB9A
SCHEMBL31389953 0.77 NPC1 (0.58) ADORA2AADORA1ALDH1A1NPC1RAB9A
SCHEMBL5565192 0.75 ADORA2A (0.83) LRRK2ADORA2AADORA1GAAMEN1
SCHEMBL22027658 0.74 ADORA2A (0.55) LRRK2ADORA2AADORA1GAAMEN1
SCHEMBL30127956 0.74 ADORA2A (0.55) LRRK2ADORA2AADORA1GAAMEN1
SCHEMBL30128220 0.74 ADORA2A (0.46) LRRK2ADORA2AADORA1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997681-B Thiazolopyridine derivatives as adenosine receptor antagonists 默克专利股份公司 2022-11-15 CN disclosed