SCHEMBL29942136

SCHEMBL29942136

Clc1ccc2cc(I)n(CC3CC3)c2n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 1/20 0.34
PIM1 P11309 2/20 0.33
PIM3 Q86V86 2/20 0.33
PIM2 Q9P1W9 2/20 0.33
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
CNR2 P34972 9/20 0.32
PDE5A O76074 2/20 0.32
PDE4A P27815 2/20 0.32
PDE4B Q07343 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
KCNH2 Q12809 1/20 0.32
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30
GRM2 Q14416 1/20 0.30
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
CCND2 P30279 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23755703 1.00 CCR9 (0.34) CCR9PIM1PIM3PIM2CTSL
SCHEMBL30122584 0.97 CCR9 (0.33) CCR9PIM1PIM3PIM2CTSL
SCHEMBL23777027 0.82 NOTUM (0.40) CCR9CTSLCTSSCTSKCNR2
SCHEMBL29641062 0.79 CTSL (0.38) CCR9PIM1PIM3PIM2CTSL
SCHEMBL24571978 0.79 CTSL (0.38) CCR9PIM1PIM3PIM2CTSL
SCHEMBL23756782 0.78 CCR9 (0.35) CCR9CTSLCTSSCTSKCNR2
SCHEMBL30122542 0.78 CCR9 (0.35) CCR9CTSLCTSSCTSKCNR2
SCHEMBL23755776 0.78 CCR9 (0.35) CCR9CTSLCTSSCTSKCNR2
SCHEMBL29641117 0.78 CCR9 (0.35) CCR9CTSLCTSSCTSKCNR2
SCHEMBL29850694 0.77 CCR9 (0.56) CCR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115348961-B Heterocyclic PAD4 inhibitors 百时美施贵宝公司 2025-03-04 CN disclosed
EP-4103559-A1 HETEROCYCLIC PAD4 INHIBITORS Bristol-Myers Squibb Company (US) 2022-12-21 EP disclosed
CN-115348961-A Heterocyclic PAD4 inhibitors 百时美施贵宝公司 2022-11-15 CN disclosed