SCHEMBL29945209

SCHEMBL29945209

C=CC(=O)N1CCN[C@@H](C(F)(F)F)C1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TEAD1 P28347 10/20 0.36
SCN7A Q01118 1/20 0.34
KCNH2 Q12809 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
BTK Q06187 3/20 0.32
JAK3 P52333 4/20 0.32
KRAS P01116 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27807646 0.81 KCNH2 (0.36) SCN7AKCNH2SCN5ASCN9ASCN10A
SCHEMBL2723202 0.80 KCNH2 (0.36) SCN7AKCNH2SCN5ASCN9ASCN10A
SCHEMBL26637402 0.80 KCNH2 (0.36) SCN7AKCNH2SCN5ASCN9ASCN10A
SCHEMBL22118053 0.80 KCNH2 (0.36) SCN7AKCNH2SCN5ASCN9ASCN10A
SCHEMBL15826470 0.78 KCNH2 (0.35) SCN7AKCNH2SCN5ASCN9ASCN10A
SCHEMBL14773479 0.78 CHRNB2 (0.37) SCN7AKCNH2SCN5ASCN9ASCN10A
SCHEMBL12331138 0.78 CHRNB2 (0.37) SCN7AKCNH2SCN5ASCN9ASCN10A
SCHEMBL14773537 0.78 CHRNB2 (0.37) SCN7AKCNH2SCN5ASCN9ASCN10A
Trifluoroacetic Acid SCHEMBL20296403 0.77 BIRC2 (0.36) TEAD1SCN9ASCN10ABTKJAK3
Trifluoroacetic Acid SCHEMBL20296401 0.77 BIRC2 (0.36) TEAD1SCN9ASCN10ABTKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115073450-A KRAS G12C Preparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed