SCHEMBL29947339

SCHEMBL29947339

CC(C)(C)OC(=O)N1CC=C(c2cccc(OCc3ccc(C#N)cc3F)n2)CC1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GLP1R P43220 4/20 0.47
GRM5 P41594 8/20 0.47
GRM1 Q13255 8/20 0.47
GPR119 Q8TDV5 2/20 0.45
PDE10A Q9Y233 2/20 0.43
ELANE P08246 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22391958 1.00 GLP1R (0.47) GLP1RGRM5GRM1GPR119PDE10A
SCHEMBL22932920 0.90 GPR119 (0.47) GRM5GRM1GPR119ELANE
SCHEMBL24321922 0.89 GRM1 (0.50) GRM5GRM1GPR119
SCHEMBL30583878 0.89 GRM1 (0.54) GRM5GRM1GPR119
SCHEMBL30120528 0.88 GLP1R (0.52) GLP1RPDE10A
SCHEMBL29668627 0.88 GRM1 (0.49) GLP1RGRM5GRM1GPR119
SCHEMBL24321526 0.88 GRM1 (0.49) GLP1RGRM5GRM1GPR119
SCHEMBL22933049 0.87 GPR119 (0.44) GLP1RGRM5GRM1GPR119ELANE
SCHEMBL24498578 0.87 GRM1 (0.46) GRM5GRM1GPR119ELANE
SCHEMBL29668677 0.87 GPR119 (0.44) GLP1RGRM5GRM1GPR119ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119638670-A Condensed imidazole derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2025-03-18 CN disclosed
CN-115244056-B Condensed imidazole derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2024-11-15 CN disclosed
CN-115867546-B Salt and crystalline forms of GLP-1R agonists and uses thereof 上海齐鲁锐格医药研发有限公司 2024-10-18 CN disclosed
CN-118344349-A 4-Alkoxybenzimidazole-6-carboxylic acid derivatives as GLP-1 receptor agonists 中国科学院上海药物研究所 2024-07-16 CN disclosed
CN-113801136-B Imidazo heteroaryl derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2023-04-07 CN disclosed
EP-4157832-A1 SALT AND CRYSTAL FORMS OF GLP-1R AGONISTS AND USES THEREOF Qilu Regor Therapeutics Inc. (CN) 2023-04-05 EP disclosed
CN-115867546-A Salts and crystalline forms of GLP-1R agonists and uses thereof 上海齐鲁锐格医药研发有限公司 2023-03-28 CN disclosed
CN-115244056-A Condensed imidazole derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-10-25 CN disclosed