SCHEMBL29950798

SCHEMBL29950798

O=CCc1ccc2ccoc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.56
CHRM1 P11229 2/20 0.56
CHRM3 P20309 2/20 0.56
HTR1B P28222 9/20 0.50
CYP2A6 P11509 2/20 0.43
KDM4E B2RXH2 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
NFKB1 P19838 1/20 0.42
MAOA P21397 1/20 0.42
ACHE P22303 1/20 0.42
CYP2C19 P33261 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.38
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA3 P07451 1/20 0.34
CA4 P22748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6186816 0.85 CYP2A6 (0.56) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL29952165 0.85 CYP2A6 (0.56) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL25235422 0.84 CHRM2 (0.60) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL29957913 0.84 CHRM2 (0.60) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL29017001 0.83 HTR1B (0.53) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL25240905 0.81 CHRM2 (0.62) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL29016962 0.80 HTR1B (0.51) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL11980461 0.79 CHRM2 (0.51) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL2490953 0.79 HTR1B (0.45) CHRM2CHRM1CHRM3HTR1BCYP2A6
SCHEMBL9111859 0.76 HTR1B (0.43) CHRM2CHRM1CHRM3HTR1BCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed