SCHEMBL2490953

SCHEMBL2490953

ON=CCc1ccc2ccoc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 9/20 0.45
CHRM2 P08172 2/20 0.44
CHRM1 P11229 2/20 0.44
CHRM3 P20309 2/20 0.44
MRGPRX4 Q96LA9 1/20 0.35
CYP2A6 P11509 3/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
NFKB1 P19838 1/20 0.34
MAOA P21397 1/20 0.34
ACHE P22303 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA7 P36544 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29950798 0.79 CHRM2 (0.56) HTR1BCHRM2CHRM1CHRM3MRGPRX4
SCHEMBL29017001 0.77 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3MRGPRX4
SCHEMBL29016962 0.75 HTR1B (0.51) HTR1BCHRM2CHRM1CHRM3MRGPRX4
SCHEMBL4328740 0.74 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3MRGPRX4
SCHEMBL9113003 0.74 HTR1B (0.43) HTR1BCHRM2CHRM1CHRM3MRGPRX4
SCHEMBL9111859 0.74 HTR1B (0.43) HTR1BCHRM2CHRM1CHRM3MRGPRX4
SCHEMBL8790466 0.72 KDM4E (0.48) CYP2A6KDM4E
SCHEMBL957248 0.71 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3MRGPRX4
SCHEMBL17613378 0.71 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3MRGPRX4
SCHEMBL507041 0.71 HTR1B (0.53) HTR1BCHRM2CHRM1CHRM3MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379542-A1 NOVEL OXIME DERIVATIVES Cadila Healthcare Limited (IN) 2011-10-26 EP disclosed
WO-2010084512-A1 NOVEL OXIME DERIVATIVES CADILA HEALTHCARE LIMITED (IN) 2010-07-29 WO disclosed