SCHEMBL29953780

SCHEMBL29953780

Nc1cc(C=O)c(-c2ccncc2)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.42
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
CHEK2 O96017 1/20 0.38
ALOX5AP P20292 1/20 0.37
FEN1 P39748 1/20 0.37
AURKB Q96GD4 2/20 0.36
INCENP Q9NQS7 2/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
DYRK1A Q13627 1/20 0.36
ABL1 P00519 1/20 0.36
FYN P06241 1/20 0.36
MAPT P10636 1/20 0.36
AKT1 P31749 1/20 0.35
PIK3CA P42336 1/20 0.35
NTRK1 P04629 2/20 0.35
AAK1 Q2M2I8 1/20 0.34
AURKA O14965 1/20 0.34
TTK P33981 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29955163 0.85 FGFR1 (0.47) ADORA2AADORA1ALOX5APFEN1MAP4K4
SCHEMBL29952599 0.83 ERN1 (0.52) ERN1CHEK2DYRK1AALDH1A1
SCHEMBL2562642 0.82 ALOX5AP (0.44) ADORA1ALOX5APFEN1ABL1MAPT
SCHEMBL2562852 0.81 FEN1 (0.56) ALOX5APFEN1MAP4K4
SCHEMBL31195690 0.78 ERN1 (0.53) ERN1AURKBINCENPPDE3BPDE3A
SCHEMBL2552689 0.75 ALOX5AP (0.42) CHEK2ALOX5APFEN1AURKBDYRK1A
SCHEMBL2555064 0.75 ALOX5AP (0.45) ALOX5APFEN1ABL1CCNT1CDK9
SCHEMBL2558043 0.72 ALOX5AP (0.53) ADORA2AADORA1ALOX5APFEN1MAPT
SCHEMBL30745188 0.72 ERN1 (0.66) ERN1PDE3BPDE3AMAPTPIK3CA
SCHEMBL14840544 0.72 ERN1 (0.47) ERN1MAPTALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed