SCHEMBL29952599

SCHEMBL29952599

Nc1cc(C=O)c(-c2cccnc2)cn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.52
CYP2A6 P11509 5/20 0.45
CYP3A4 P08684 4/20 0.45
CYP2E1 P05181 3/20 0.45
CYP2C9 P11712 3/20 0.45
CYP2B6 P20813 3/20 0.45
CYP2C19 P33261 3/20 0.45
DYRK1A Q13627 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
TDO2 P48775 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
PTK2 Q05397 1/20 0.43
MKNK1 Q9BUB5 2/20 0.42
MKNK2 Q9HBH9 2/20 0.42
MEN1 O00255 1/20 0.42
PSIP1 O75475 1/20 0.42
AXL P30530 1/20 0.42
PIK3C3 Q8NEB9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29955163 0.84 FGFR1 (0.47) MEN1
SCHEMBL29953780 0.83 ERN1 (0.42) ERN1DYRK1ACHEK2ALDH1A1
SCHEMBL2552689 0.78 ALOX5AP (0.42) DYRK1AMEN1CHEK2
SCHEMBL16835900 0.76 TDO2 (0.47) ERN1CYP2A6CYP3A4CYP2E1CYP2C9
SCHEMBL16826222 0.76 CYP2A6 (0.50) CYP2A6CYP3A4CYP2E1CYP2C9CYP2B6
SCHEMBL28494615 0.76 KMO (0.49) DYRK1ADYRK1BMKNK1MKNK2MEN1
SCHEMBL2562642 0.75 ALOX5AP (0.44) CYP3A4TDO2MEN1ALDH1A1CYP1A2
SCHEMBL1802008 0.75 ERN1 (0.59) ERN1CYP2A6CYP3A4CYP2E1CYP2C9
SCHEMBL2558043 0.74 ALOX5AP (0.53) MEN1ALDH1A1
SCHEMBL17009195 0.74 ERN1 (0.54) ERN1CYP2A6CYP3A4CYP2E1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed