SCHEMBL29955947

SCHEMBL29955947

OB(O)c1cc2ccccc2nc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.50
ALDH1A1 P00352 6/20 0.46
HPGD P15428 2/20 0.46
GLA P06280 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
MAPT P10636 2/20 0.46
ACHE P22303 1/20 0.46
KDM4E B2RXH2 5/20 0.44
GAA P10253 2/20 0.44
STAT3 P40763 1/20 0.44
EGFR P00533 1/20 0.42
TOP2A P11388 1/20 0.42
TOP2B Q02880 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
ALOX5 P09917 2/20 0.38
HTT P42858 2/20 0.38
PDE10A Q9Y233 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HTR3B O95264 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL115832 1.00 KMT2A (0.50) KMT2AALDH1A1HPGDGLATDP1
SCHEMBL1670726 0.89 KMT2A (0.41) KMT2AALDH1A1HPGDGLATDP1
SCHEMBL29951444 0.78 ALDH1A1 (0.48) KMT2AALDH1A1HPGDGLATDP1
SCHEMBL16488132 0.78 ALDH1A1 (0.60) KMT2AALDH1A1HPGDGLATDP1
SCHEMBL789653 0.78 ALDH1A1 (0.48) KMT2AALDH1A1HPGDGLATDP1
SCHEMBL29955400 0.78 ALDH1A1 (0.50) KMT2AALDH1A1HPGDGLATDP1
SCHEMBL2074966 0.78 ALDH1A1 (0.46) KMT2AALDH1A1HPGDGLAMAPT
SCHEMBL29955290 0.78 ALDH1A1 (0.46) KMT2AALDH1A1HPGDGLAMAPT
SCHEMBL2717631 0.77 PDE3B (0.42) KMT2ATDP1MAPTKDM4EEGFR
SCHEMBL14012754 0.77 MAP4K4 (0.33) ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119677737-A Heteroaryl compounds for the treatment of pain 沃泰克斯药物股份有限公司 2025-03-21 CN disclosed
CN-119546580-A Heteroaryl compounds for the treatment of pain 沃泰克斯药物股份有限公司 2025-02-28 CN disclosed
EP-4511116-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN Vertex Pharmaceuticals Incorporated (US) 2025-02-26 EP disclosed
EP-4511115-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN Vertex Pharmaceuticals Incorporated (US) 2025-02-26 EP disclosed
WO-2023205468-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-10-26 WO disclosed
WO-2023205463-A1 HETEROARYL COMPOUNDS FOR THE TREATMENT OF PAIN VERTEX PHARMACEUTICALS INCORPORATED (US) 2023-10-26 WO disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed