SCHEMBL29956067

SCHEMBL29956067

CC(C)(C)OC(=O)Nc1ccc(B(O)O)cc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.50
KCNQ4 P56696 3/20 0.41
KCNQ5 Q9NR82 3/20 0.41
RXFP1 Q9HBX9 1/20 0.39
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA9 Q16790 1/20 0.37
HTT P42858 1/20 0.37
HIF1A Q16665 1/20 0.37
METAP1 P53582 1/20 0.37
ESR1 P03372 1/20 0.37
ESRRG P62508 1/20 0.37
ESR2 Q92731 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
BRD9 Q9H8M2 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1256341 1.00 CYP17A1 (0.50) CYP17A1KCNQ4KCNQ5RXFP1CA12
SCHEMBL3784938 0.87 HPGD (0.44) CYP17A1KCNQ4KCNQ5RXFP1CA12
SCHEMBL21682754 0.84 SMN1; SMN2 (0.44) CYP17A1KCNQ4KCNQ5RXFP1CA12
SCHEMBL857284 0.82 HTT (0.55) CYP17A1KCNQ4KCNQ5HTTLMNA
SCHEMBL15925258 0.82 CYP17A1 (0.54) CYP17A1KCNQ4KCNQ5RXFP1CA12
SCHEMBL169631 0.82 HTT (0.44) HTTLMNAPOLBNPSR1
SCHEMBL29952945 0.81 LMNA (0.41) RXFP1CA12CA1CA9HIF1A
SCHEMBL2363945 0.81 CYP17A1 (0.53) CYP17A1KCNQ4KCNQ5RXFP1HTT
SCHEMBL29834708 0.81 CYP17A1 (0.53) CYP17A1KCNQ4KCNQ5RXFP1HTT
SCHEMBL6134887 0.81 ATR (0.45) CYP17A1RXFP1CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119301105-A Thiostrepton-based compounds for the treatment of cancer and preparation thereof RS肿瘤学有限责任公司 2025-01-10 CN disclosed
WO-2024131893-A1 IRE1α SMALL MOLECULE INHIBITORS SHANGHAI YI ZHONG XING BIOTECHNOLOGY CO., LTD. (CN) 2024-06-27 WO disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed