SCHEMBL29956460

SCHEMBL29956460

O=Cc1ccnc2[nH]cc(I)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.47
CHEK1 O14757 2/20 0.42
CCR1 P32246 1/20 0.39
CCR5 P51681 1/20 0.39
CCR8 P51685 1/20 0.39
LRRK2 Q5S007 6/20 0.35
ROCK2 O75116 5/20 0.33
ROCK1 Q13464 5/20 0.33
CDC42BPA Q5VT25 4/20 0.33
CDC42BPB Q9Y5S2 4/20 0.33
TRPA1 O75762 1/20 0.33
CDK9 P50750 3/20 0.32
CDK2 P24941 2/20 0.32
CDK5 Q00535 2/20 0.32
CDC7 O00311 1/20 0.32
PLK4 O00444 1/20 0.32
MAPK13 O15264 1/20 0.32
PDPK1 O15530 1/20 0.32
DAPK3 O43293 1/20 0.32
DYRK3 O43781 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29952688 0.86 KMT2A (0.51) KMT2ACHEK1CCR1CCR5CCR8
SCHEMBL29957196 0.84 KMT2A (0.56) KMT2ACHEK1CCR1CCR5CCR8
SCHEMBL21428928 0.81 KMT2A (0.49) KMT2ACHEK1CCR1CCR5CCR8
SCHEMBL29935820 0.81 KMT2A (0.49) KMT2ACHEK1CCR1CCR5CCR8
SCHEMBL29953901 0.79 KMT2A (0.47) KMT2ACHEK1CCR1CCR5CCR8
SCHEMBL29958532 0.79 KMT2A (0.47) KMT2ACHEK1CCR1CCR5CCR8
SCHEMBL26176313 0.77 CHEK1 (0.46) CHEK1LRRK2ROCK2ROCK1CDC42BPA
SCHEMBL29952435 0.76 LRRK2 (0.51) KMT2ACHEK1LRRK2ROCK2ROCK1
SCHEMBL16854295 0.75 CHEK1 (0.49) KMT2ACHEK1TRPA1AXLMAPK1
SCHEMBL29955671 0.74 KMT2A (0.43) KMT2ACCR1CCR5CCR8LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed