SCHEMBL29957539

SCHEMBL29957539

O=Cc1cccc2[nH]cc(Br)c12

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.74
IMPDH2 P12268 1/20 0.47
PIM1 P11309 3/20 0.47
PIM3 Q86V86 3/20 0.47
PIM2 Q9P1W9 2/20 0.47
ERN1 O75460 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
THRB P10828 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TRIM24 O15164 2/20 0.36
TRIM33 Q9UPN9 2/20 0.36
CLK1 P49759 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
GPR84 Q9NQS5 3/20 0.33
FFAR1 O14842 1/20 0.33
AHR P35869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29953853 0.85 CYP2A6 (1.00) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL644301 0.85 CYP2A6 (1.00) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL29952428 0.82 CYP2A6 (0.70) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL29951403 0.78 CYP2A6 (0.54) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL15672105 0.78 CYP2A6 (0.54) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL31279438 0.78 CYP2A6 (0.54) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL7327866 0.78 CYP2A6 (0.54) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL27308948 0.78 CYP2A6 (0.54) CYP2A6IMPDH2PIM1PIM3PIM2
SCHEMBL28973447 0.76 CYP2A6 (0.60) CYP2A6PIM1PIM3PIM2CLK1
SCHEMBL248842 0.72 CYP2A6 (0.66) CYP2A6IMPDH2PIM1PIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed