SCHEMBL29958145

SCHEMBL29958145

O=Cc1ccc(C2CNC2)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.35
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
F2R P25116 1/20 0.32
CCR1 P32246 1/20 0.31
CHRNB4 P30926 2/20 0.31
CHRNA3 P32297 2/20 0.31
HTR3A P46098 2/20 0.30
CHRNA1 P02708 1/20 0.30
ESR1 P03372 1/20 0.30
CHRNG P07510 1/20 0.30
CHRNB1 P11230 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29955701 0.87 HTR3A (0.47) DDB1CRBNHTR3A
SCHEMBL29952339 0.85
SCHEMBL21355057 0.83 KDM4E (0.42) KCNJ1DDB1CRBNKDM4EGLA
SCHEMBL32684974 0.83 KDM4E (0.42) KCNJ1DDB1CRBNKDM4EGLA
SCHEMBL29951949 0.83 DDB1 (0.47) DDB1CRBNKDM4EGLAHTT
SCHEMBL26817536 0.81 HTT (0.49) KCNJ1DDB1CRBNKDM4EGLA
SCHEMBL2559816 0.77 PARP1 (0.33) KCNJ1
SCHEMBL2562746 0.77 PARP1 (0.33) KCNJ1
SCHEMBL24666229 0.76 KCNJ1 (0.33) KCNJ1KDM4EGLAHTTKMT2A
SCHEMBL24323731 0.76 F2R (0.38) KCNJ1KDM4EGLAHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed