SCHEMBL29960002

SCHEMBL29960002

CCCCOC(=O)c1ccc(CN2C(=O)c3ccccc3C2=O)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.58
ALDH1A1 P00352 4/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.56
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
TSHR P16473 4/20 0.54
LMNA P02545 4/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2C19 P33261 2/20 0.54
MAPK1 P28482 2/20 0.54
ESR1 P03372 1/20 0.54
CYP2D6 P10635 1/20 0.54
NR1H2 P55055 1/20 0.54
RNASEL Q05823 1/20 0.54
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
PDE4D Q08499 1/20 0.52
CASP3 P42574 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL916911 0.87 KMT2A (0.65) GAAALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL3664093 0.85 TSHR (0.55) ALDH1A1TSHRLMNAMAPK1CYP3A4
SCHEMBL14597968 0.81 HDAC1 (0.67) MEN1KMT2AHDAC1HDAC7MAPK1
SCHEMBL10766110 0.81 SMN1; SMN2 (0.64) GAAALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL6318770 0.77 HDAC1 (0.58) ALDH1A1MEN1KMT2AHDAC1HDAC7
SCHEMBL10988558 0.77 ESR1 (0.74) GAAALDH1A1SMN1; SMN2TSHRLMNA
SCHEMBL37476 0.77 ESR1 (0.85) GAAALDH1A1SMN1; SMN2TSHRLMNA
SCHEMBL8084590 0.76 TSHR (0.64) ALDH1A1SMN1; SMN2TSHRLMNACYP1A2
SCHEMBL28816311 0.76 SMN1; SMN2 (0.66) GAAALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL12905303 0.76 HDAC1 (0.68) ALDH1A1MEN1KMT2AHDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4065572-A1 BENZYLAMIDE DERIVATIVES AS INHIBITORS OF TRANSFORMING GROWTH FACTOR-BETA RECEPTOR I/ALK5 Origo Biopharma, S.L. (ES) 2022-10-05 EP disclosed