Predicted protein targets (top 19)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | HCAR3 | P49019 | 9/20 | 0.50 |
| ▸ | KDM4E | B2RXH2 | 3/20 | 0.50 |
| ▸ | HPGD | P15428 | 4/20 | 0.44 |
| ▸ | ALDH1A1 | P00352 | 2/20 | 0.44 |
| ▸ | CPT2 | P23786 | 1/20 | 0.43 |
| ▸ | CPT1A | P50416 | 1/20 | 0.43 |
| ▸ | CPT1B | Q92523 | 1/20 | 0.43 |
| ▸ | GRIN2D | O15399 | 1/20 | 0.43 |
| ▸ | GRIN2A | Q12879 | 1/20 | 0.43 |
| ▸ | GRIN2C | Q14957 | 1/20 | 0.43 |
| ▸ | TEAD1 | P28347 | 1/20 | 0.41 |
| ▸ | TEAD4 | Q15561 | 1/20 | 0.41 |
| ▸ | TEAD2 | Q15562 | 1/20 | 0.41 |
| ▸ | TEAD3 | Q99594 | 1/20 | 0.41 |
| ▸ | HCAR2 | Q8TDS4 | 1/20 | 0.40 |
| ▸ | TBXAS1 | P24557 | 1/20 | 0.40 |
| ▸ | RORC | P51449 | 1/20 | 0.39 |
| ▸ | TSHR | P16473 | 1/20 | 0.39 |
| ▸ | HSD17B10 | Q99714 | 1/20 | 0.39 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL121802 | 0.87 | SLC2A1 (0.41) | HCAR3KDM4EHPGDALDH1A1CPT2 | |
| SCHEMBL14737303 | 0.83 | MAPT (0.50) | KDM4EHPGDALDH1A1TSHRHSD17B10 | |
| SCHEMBL31173872 | 0.83 | MAPT (0.50) | KDM4EHPGDALDH1A1TSHRHSD17B10 | |
| SCHEMBL23535727 | 0.82 | HCAR3 (0.55) | HCAR3KDM4EHPGDALDH1A1CPT2 | |
| SCHEMBL30040739 | 0.82 | HCAR3 (0.55) | HCAR3KDM4EHPGDALDH1A1CPT2 | |
| SCHEMBL14869360 | 0.81 | HCAR3 (0.50) | HCAR3KDM4EHPGDALDH1A1CPT2 | |
| SCHEMBL25113848 | 0.81 | HCAR3 (0.50) | HCAR3KDM4EHPGDALDH1A1CPT2 | |
| SCHEMBL23559718 | 0.81 | HCAR3 (0.50) | HCAR3KDM4EHPGDALDH1A1CPT2 | |
| SCHEMBL30189248 | 0.81 | HCAR3 (0.50) | HCAR3KDM4EHPGDALDH1A1CPT2 | |
| SCHEMBL29301488 | 0.81 | HCAR3 (0.50) | HCAR3KDM4EHPGDALDH1A1CPT2 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| WO-2022159454-A1 | BET SUBFAMILY INHIBITORS AND METHODS USING SAME | BAYLOR COLLEGE OF MEDICINE (US) | 2022-07-28 | — | — | WO | disclosed |