SCHEMBL29960424

SCHEMBL29960424

c1cncc(-c2cccc3[nH]cnc23)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 1/20 0.51
QPCTL Q9NXS2 1/20 0.51
BRD4 O60885 2/20 0.50
DYRK1A Q13627 3/20 0.46
GSK3B P49841 1/20 0.46
MAPK1 P28482 1/20 0.46
NUDT1 P36639 1/20 0.45
CYP2A6 P11509 3/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2E1 P05181 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2B6 P20813 1/20 0.45
CYP2C19 P33261 1/20 0.45
CLK2 P49760 2/20 0.44
CLK3 P49761 2/20 0.44
WNT1 P04628 1/20 0.44
TGFBR1 P36897 1/20 0.44
PARP1 P09874 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27143869 1.00 QPCT (0.51) QPCTQPCTLBRD4DYRK1AGSK3B
SCHEMBL31501287 0.90 BRD4 (0.49) QPCTQPCTLBRD4DYRK1AGSK3B
SCHEMBL903206 0.83 BRD4 (0.52) QPCTQPCTLBRD4MAPK1CLK2
SCHEMBL29477064 0.81 DPP4 (0.57) BRD4CYP3A4PARP1ALDH1A1ABL1
SCHEMBL3858256 0.81 DPP4 (0.57) BRD4CYP3A4PARP1ALDH1A1ABL1
SCHEMBL20878376 0.78 BRD4 (0.56) BRD4PARP1ALDH1A1ABL1
SCHEMBL21744628 0.77 TDO2 (0.56) QPCTQPCTLBRD4DYRK1AGSK3B
SCHEMBL28094392 0.77 BRD4 (0.52) QPCTQPCTLBRD4DYRK1AMAPK1
SCHEMBL903194 0.75 CYP17A1 (0.50) BRD4CYP1A2TDO2
SCHEMBL900109 0.75 CYP17A1 (0.48) QPCTQPCTLBRD4DYRK1AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4326723-A1 PYRIMIDO[5,4,D]PYRIMIDINE COMPOUNDS, COMPOSITIONS COMPRISING THEM AND USES THEREOF Université de Montréal (CA) 2024-02-28 EP disclosed
WO-2022221940-A1 PYRIMIDO[5,4,D]PYRIMIDINE COMPOUNDS, COMPOSITIONS COMPRISING THEM AND USES THEREOF UNIVERSITE DE MONTREAL (CA) 2022-10-27 WO disclosed