SCHEMBL29960862

SCHEMBL29960862

Cc1cc2ncc(CBr)cc2[nH]c1=O

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 1/20 0.50
PARP1 P09874 17/20 0.45
PARP2 Q9UGN5 2/20 0.37
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29115637 1.00 ATAD2 (0.50) ATAD2PARP1PARP2BRD4
SCHEMBL25606713 0.86 ATAD2 (0.51) ATAD2PARP1PARP2
SCHEMBL25604620 0.84 ATAD2 (0.50) ATAD2PARP1PARP2BRD4
SCHEMBL25606715 0.84 ATAD2 (0.50) ATAD2PARP1PARP2BRD4
SCHEMBL25604619 0.84 ATAD2 (0.50) ATAD2PARP1PARP2
SCHEMBL30331559 0.84 ATAD2 (0.50) ATAD2PARP1PARP2
SCHEMBL30663279 0.84 ATAD2 (0.50) ATAD2PARP1PARP2BRD4
SCHEMBL29396473 0.83 PARP1 (0.52) PARP1PARP2
SCHEMBL22912684 0.83 PARP1 (0.52) PARP1PARP2
SCHEMBL29960664 0.81 PARP1 (0.45) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710433-A Selective PARP1 inhibitor and application thereof 成都百裕制药股份有限公司 2023-09-05 CN disclosed
WO-2022222966-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2022-10-27 WO disclosed