SCHEMBL29960965

SCHEMBL29960965

NC(=O)c1ccc(N2CCNCC2)cc1CCO

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 6/20 0.50
TGFBR1 P36897 2/20 0.45
AOC3 Q16853 1/20 0.42
ADRB1 P08588 3/20 0.41
ALDH1A1 P00352 2/20 0.40
USP2 O75604 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
HTR3E A5X5Y0 2/20 0.40
HTR3B O95264 2/20 0.40
HTR3A P46098 2/20 0.40
HTR3D Q70Z44 2/20 0.40
HTR3C Q8WXA8 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29115599 0.97 ACVR1 (0.48) ACVR1TGFBR1AOC3ADRB1ALDH1A1
SCHEMBL29960909 0.85 ACVR1 (0.54) ACVR1TGFBR1AOC3ADRB1CHRNB2
SCHEMBL29115436 0.83 ACVR1 (0.52) ACVR1TGFBR1AOC3ADRB1CHRNB2
SCHEMBL30879569 0.79 MAPT (0.55) ACVR1TGFBR1ADRB1ALDH1A1USP2
SCHEMBL3633976 0.77 ACVR1 (0.62) ACVR1TGFBR1ADRB1ALDH1A1USP2
SCHEMBL1741562 0.77 ADRB1 (0.61) ACVR1TGFBR1ADRB1ALDH1A1USP2
SCHEMBL30798753 0.77 ADRB1 (0.61) ACVR1TGFBR1ADRB1ALDH1A1USP2
Hydrochloric Acid SCHEMBL27825221 0.76 ACVR1 (0.61) ACVR1TGFBR1ADRB1ALDH1A1USP2
SCHEMBL1598681 0.76 ADRB1 (0.46) AOC3ADRB1ALDH1A1CHRNB2CHRNA4
SCHEMBL29138207 0.74 ADRB1 (0.61) ACVR1TGFBR1ADRB1ALDH1A1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710433-A Selective PARP1 inhibitor and application thereof 成都百裕制药股份有限公司 2023-09-05 CN disclosed
WO-2022222966-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2022-10-27 WO disclosed