SCHEMBL29966673

SCHEMBL29966673

CC(=Cc1ccc(C(F)(F)F)nc1)C(=O)Nc1ccccc1C(=O)O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.64
TRPM8 Q7Z2W7 3/20 0.64
TRPA1 O75762 4/20 0.46
TAS2R14 Q9NYV8 3/20 0.44
MAPK1 P28482 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
STAT1 P42224 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TRPM2 O94759 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21470183 1.00 DHODH (0.64) DHODHTRPM8TRPA1TAS2R14MAPK1
SCHEMBL8048868 0.82 TRPM8 (0.76) DHODHTRPM8TRPA1TAS2R14TRPM2
SCHEMBL8048873 0.82 TRPM8 (0.76) DHODHTRPM8TRPA1TAS2R14TRPM2
SCHEMBL29966740 0.82 TRPM8 (0.76) DHODHTRPM8TRPA1TAS2R14TRPM2
Lithium SCHEMBL8048874 0.81 TRPM8 (0.74) DHODHTRPM8TRPA1TAS2R14TRPM2
SCHEMBL8058714 0.81 TRPM8 (0.74) DHODHTRPM8TRPA1TAS2R14ALDH1A1
SCHEMBL8060378 0.81 TRPM8 (0.74) DHODHTRPM8TRPA1TAS2R14TRPM2
SCHEMBL8060371 0.81 TRPM8 (0.74) DHODHTRPM8TRPA1TAS2R14TRPM2
SCHEMBL8065731 0.79 DHODH (1.00) DHODHTRPM8TRPA1NPC1RAB9A
SCHEMBL8065734 0.79 DHODH (1.00) DHODHTRPM8TRPA1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110357789-B N-substituted acrylamide derivative as DHODH inhibitor and preparation and application thereof 华东理工大学 2022-09-30 CN disclosed