SCHEMBL29967017

SCHEMBL29967017

COC(=O)CC[C@@H]1C[C@H](c2c(OC)ccc(Cl)c2Cl)CN1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.41
HTR2C P28335 6/20 0.41
HTR2B P41595 5/20 0.41
DRD2 P14416 2/20 0.36
TNF P01375 2/20 0.34
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
PDE4B Q07343 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23217313 1.00 HTR2A (0.41) HTR2AHTR2CHTR2BDRD2TNF
SCHEMBL23217292 0.90 HTR2A (0.38) HTR2AHTR2CHTR2BDRD2TNF
SCHEMBL23217451 0.88 HTR2A (0.40) HTR2AHTR2CHTR2BDRD2TNF
SCHEMBL25034602 0.87 HTR2A (0.40) HTR2AHTR2CHTR2BDRD2TNF
SCHEMBL23217435 0.85 HTR2C (0.45) HTR2AHTR2CHTR2BDRD2KMT2A
SCHEMBL23217075 0.84 HTR2A (0.47) HTR2AHTR2CHTR2BDRD2KMT2A
SCHEMBL23217276 0.83 HTR2A (0.35) HTR2AHTR2CHTR2BDRD2
SCHEMBL23217775 0.83 HTR2A (0.43) HTR2AHTR2CHTR2BDRD2KMT2A
SCHEMBL23217362 0.82 HTR2A (0.42) HTR2AHTR2CHTR2BDRD2KMT2A
SCHEMBL23217543 0.82 HTR2A (0.42) HTR2AHTR2CHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114828963-A Arylheterobicyclic compounds as Kv1.3 potassium SHAKER channel blockers D·E·萧尔研究有限责任公司 2022-07-29 CN disclosed