SCHEMBL29967682

SCHEMBL29967682

CC(C)c1nc2c(-c3ccc(C4=CCCCC4)cc3)cccc2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.39
PSMB5 P28074 3/20 0.36
HSD17B10 Q99714 2/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
PARP1 P09874 5/20 0.34
KDM5B Q9UGL1 1/20 0.34
FFAR2 O15552 1/20 0.33
TRPV3 Q8NET8 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
ADORA1 P30542 1/20 0.32
CNR2 P34972 3/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29967926 0.84 PTGS2 (0.41) PTGS2PSMB5PARP1FFAR2CNR2
SCHEMBL29968177 0.81 PTGS2 (0.39) PTGS2PSMB5HSD17B10FFAR2ADORA3
SCHEMBL29968000 0.79 DHODH (0.48) PTGS2PARP1CNR2
SCHEMBL12960725 0.79 KDM4E (0.43) HSD17B10KDM4ELMNAALDH1A1HPGD
SCHEMBL29967779 0.79 PTGS2 (0.38) PTGS2PSMB5PARP1FFAR2ADORA3
SCHEMBL29968037 0.78 PARP1 (0.39) KDM4EALDH1A1HPGDPARP1CNR2
SCHEMBL29967862 0.77 PIK3CD (0.37) PTGS2FFAR2CNR2
SCHEMBL29968235 0.77 PSMB5 (0.41) PTGS2PSMB5PARP1
SCHEMBL29967810 0.76 PIK3CD (0.37) PTGS2PARP1FFAR2CNR2
SCHEMBL29967941 0.75 PIK3CD (0.36) PTGS2PARP1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed