SCHEMBL29967702

SCHEMBL29967702

Nc1nn(CCO)c2cccc(-c3ccc(Br)cc3)c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.56
FLT3 P36888 6/20 0.56
LCK P06239 2/20 0.46
CSF1R P07333 2/20 0.46
PLK4 O00444 1/20 0.46
AURKA O14965 1/20 0.46
JAK2 O60674 1/20 0.46
CDK1 P06493 1/20 0.46
LYN P07948 1/20 0.46
FGFR1 P11362 1/20 0.46
SRC P12931 1/20 0.46
PRKACA P17612 1/20 0.46
RPS6KB1 P23443 1/20 0.46
CDK2 P24941 1/20 0.46
MARK3 P27448 1/20 0.46
AKT1 P31749 1/20 0.46
AKT2 P31751 1/20 0.46
BLK P51451 1/20 0.46
CSNK2A1 P68400 1/20 0.46
ROCK1 Q13464 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28871292 1.00 KDR (0.56) KDRFLT3LCKCSF1RPLK4
SCHEMBL29967807 0.79 KDR (0.50) KDRFLT3LCKCSF1RAKT1
SCHEMBL29968393 0.75 KDR (0.45) KDRFLT3SCN5ASCN9AGAA
SCHEMBL28871294 0.75 KDR (0.45) KDRFLT3SCN5ASCN9AGAA
SCHEMBL419499 0.73 KDR (0.56) KDRFLT3LCKCSF1RSCN5A
SCHEMBL20481783 0.71 PDGFRA (0.52) KDRFLT3JAK2CDK2SCN5A
SCHEMBL17045395 0.69 SCN9A (0.46) KDRFLT3SCN5ASCN9AMEN1
SCHEMBL422378 0.69 KDR (0.56) KDRFLT3LCKCSF1RPLK4
SCHEMBL29794328 0.68 MAPT (0.61) MEN1GALR3GAAMAPTNPY1R
SCHEMBL11120339 0.65 EIF2AK2 (0.62) KDRFLT3LCKCSF1RPLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed