SCHEMBL29967807

SCHEMBL29967807

Nc1nn(CCO)c2cccc(-c3ccc(C4=CCCCC4)cc3)c12

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.50
FLT3 P36888 5/20 0.50
SCN5A Q14524 2/20 0.35
SCN9A Q15858 2/20 0.35
PTGS2 P35354 1/20 0.35
LCK P06239 1/20 0.34
CSF1R P07333 1/20 0.34
KIT P10721 1/20 0.34
FLT1 P17948 1/20 0.34
FLT4 P35916 1/20 0.34
HDAC1 Q13547 5/20 0.33
HDAC2 Q92769 5/20 0.33
HDAC3 O15379 2/20 0.33
ACMSD Q8TDX5 1/20 0.32
TBK1 Q9UHD2 2/20 0.31
MAPK1 P28482 1/20 0.31
IKBKE Q14164 1/20 0.31
AKT1 P31749 1/20 0.30
AKT2 P31751 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29967702 0.79 KDR (0.56) KDRFLT3SCN5ASCN9ALCK
SCHEMBL28871292 0.79 KDR (0.56) KDRFLT3SCN5ASCN9ALCK
SCHEMBL29967987 0.78 MEN1 (0.37) KDRFLT3PTGS2LCKCSF1R
SCHEMBL29967634 0.75 KDR (0.38) KDRFLT3ACMSD
SCHEMBL29967871 0.75 BTK (0.38) KDRFLT3PTGS2LCKCSF1R
SCHEMBL29968082 0.69 KDR (0.63) KDRFLT3LCKCSF1RKIT
SCHEMBL28871294 0.69 KDR (0.45) KDRFLT3SCN5ASCN9AMAPK1
SCHEMBL29968393 0.69 KDR (0.45) KDRFLT3SCN5ASCN9AMAPK1
SCHEMBL12374175 0.68 KCNH2 (0.36) PTGS2HDAC1HDAC2HDAC3ACMSD
SCHEMBL419499 0.67 KDR (0.56) KDRFLT3SCN5ASCN9ALCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed